Cardarine: The Truth about GW-501516

Cardarine, better known as the GW-501516, is a supposed miracle drug that boosts immunity, endurance and burns fat. If you have just heard about GW501516, this is going to be a great learning experience for you.  We’re going to cover all important aspects of Cardarine (GW-501516) in this article.

Let the facts shine on you.

The Invention of GW501516

The invention and later transition of Cardarine are a compilation of some interesting events. It started with scientists looking for a remedy to compensate for our lifestyle. We’re talking about lifestyle that leads to diseases like heart failure, diabetes, and inflammation.

But the studies were canceled because the tested mice were found to have been diagnosed with cancer.

The invention of Cardarine (GW-501516) was possible because the scientists were looking for a PPAR-delta pathway. Why? It was because they were looking to increase physical endurance and fat burning at the same time. Once activated, the PPAR-delta pathway improves our endurance, muscle growth and fat burning characteristics dramatically.

GW501516 is one of the few discovered elements that can actively bind itself to the PPAR-delta pathway in our muscles.

The Legal Aspect of Cardarine

With the instant energy and endurance increasing capabilities of GW-501516, it’s a valid question whether it is legal or not. Unfortunately, it is not. It’s not even approved for human usage.

The possible side effects were downplayed on various forums on the internet which led to the huge popularity of Cardarine among bodybuilders and athletes. With that said, it’s now very easy to get in the black markets.

The World-Anti Doping Agency has gone one step further in its operations and issued a warning regarding the health risks of GW501516 for both the athletes and the potential ‘cheats’.

How Does Cardarine Work?

Cardarine is a PPAR agonist. PPAR is an active compound in our body that activates the androgen receptors of our muscles. It’s similar to SARMs (Selective Androgen Receptor Modulators), but it’s not.

When these receptors are activated, they increase glucose and amino acid uptake into our muscle by increasing the insulin sensitivity. GLUT-4 receptors are responsible for letting the glucose enter our cells through the cell surface membrane.

The excess amount of amino acids leads to more proteins to be synthesized. The immediate result is muscle growth and hypertrophy. In simple words, the food we eat isn’t going to be stored as fat or carbohydrate. Instead, it’s going to be stored as lean muscle mass.

Cardarine or GW-501516 also increases the level of HDL and decreases LDL. HDL is known as the good cholesterol and LDL is the bad cholesterol. Cardarine transfers HDL from the periphery to liver for metabolism purposes.

All these actions inside our body finally result in fat burn, increased endurance, and fast muscle growth.

 The working procedure of GW501516 is fairly complex and not suitable for the mass audience to understand. So, we’re not going into the details.

But, the important aspect is the benefits and side effects of Cardarine. So, people can educate themselves on GW-5015016 and decide for themselves whether to use it or not.

Benefits of Cardarine

Despite being not approved by any health organizations, Cardarine has managed to gain huge popularity for its benefits. Let’s take a look at some of them.

It Burns Fat

As Cardarine binds itself with the PPAR-delta pathway, it helps with burning fat fast. The PPAR-delta can activate quite a lot of fat-burning genes. A study was conducted on humans not too long ago to certify these claims by GW501516 users.

In that study, 13 people who were subject to excess belly fat and bad cholesterol, participated. They were given a dosage of 2.5 milligrams every day for six weeks. The results indicated that the participants dramatically reduced their cholesterol level, triglycerides, and APOB.

It Protects the Brain

Cardarine helps maintain blood flow to the brain. An animal study showed that Cardarine protects brain vessels from stress and oxidative damage.

PPAR activators are famous for their nerve cell developing properties with the help of PPAR-delta pathways.

It Helps with Obesity

Cardarine can enhance our metabolic characteristics. Hence, it works well with obesity. Study on six volunteers who suffered from obesity showed that Cardarine can reverse all metabolic syndrome without any side effects.

The participants received 2.5 to 10 milligrams of Cardarine every day for 14 days. The results were reduced liver fat, blood fat levels, and insulin. Also, GW-501516 helped to block inflammatory substances by traveling through the PPAR-delta pathways.

Also, Cardarine or GW-501516 release pro-inflammatory mediators that halt the synthesis of fatty acid. In other words, your body won’t store any fats.

How To Use Cardarine

Dosage

As we already mentioned, Cardarine is not an approved drug, so, there is no actual recommended dosage. But the most common usage is 10-20 milligrams per day for 8-12 weeks with breaks for 4-6 weeks. GW-501516 works great with other SARMs, though it’s not a SARM itself.

Usage

With so many supposed good things about Cardarine, it has gained fame across a multitude of industries. The sports industry and the fitness industry are only to name a few.

The Sports Industry

Cardarine is best known for its endurance enhancing effects. It’s common knowledge that athletes and professional sports players can gain significant results from Cardarine. It allows for more oxygen usage and promotes muscle hypertrophy and growth. The process comes with a boost in performance and stamina.

The Fitness Industry

People with strict fitness goals often fail despite being very careful with their diet and exercise, but metabolism probably has a better hand over anything else when it comes to fitness.

So, the bodybuilders who are not able to shed extra calories due to their poor metabolism can benefit vastly from Cardarine. They could expect an increase of Lipolysis without any catabolic effects. In simple words, proper preservation of lean muscle mass.

Final Thoughts

Cardarine or GW-501516, however you like to call it, comes with important health benefits. The initial studies were halted due to its cancer-causing properties in mice. But despite the risks, GW501516 has continued to be a popular drug among bodybuilders and athletes. If you decide to use it, be careful about the dosage and look for adverse effects on your health.